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奥格列汀杂质 奥格列汀异构体对照品
点击次数:1054 更新时间:2017-07-18

      奥格列汀市场前景:奥格列汀为超长效二肽基肽酶-4(DPP-4)抑制剂,其作用机制是通过抑制体内DPP-4酶对胰高血糖素样肽-1(GLP-1)的降解作用,延长GLP-1的作用时间,从而提高血液中内源性GLP-1和GIP的浓度,并zui终改善血糖控制。2013年抗糖尿病治疗药物销售额达到了469亿美元的市场规模 ,其中DPP-4抑制剂销售市场达到93.88亿美元,同比上一年增长了10.24%,是快速发展的一类药物。

 

      深圳远扬化学可提供奥格列汀申报所用全套杂质, 随货附CoA证书,HNMR,MS,HPLC图谱,纯度符合申报要求,欢迎我司(何 ;phastandards; )。请点击本页标题下方“进入该公司展台” 查看我司信息。

 

MK-3102(2R,3S,5R)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 1tert-butyl ((2S,3S)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate
MK-3102 Impurity 2tert-butyl ((2S,3R)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate
MK-3102 Impurity 3tert-butyl ((2R,3R)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate compound with tert-butyl ((2S,3S)-2-(2,5-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate (1:1)
MK-3102 Impurity 4tert-butyl ((2R,3S)-2-(2,3-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate
MK-3102 Impurity 5tert-butyl ((2R,3S)-2-(3,4-difluorophenyl)-5-oxotetrahydro-2H-pyran-3-yl)carbamate
MK-3102 Impurity 61-(methylsulfonyl)-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole
MK-3102 Impurity 7S,5R)-2-(2,5-difluorophenyl)-5-(1-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(1H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 8(2R,3S,5S)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 9(2S,3S,5S)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 10(2S,3S,5R)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 11(2S,3R,5S)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 12(2R,3R,5R)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 13(2S,3R,5R)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 14(2R,3R,5S)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 15(2R,3S,5R)-2-(2,5-difluorophenyl)-5-(pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
MK-3102 Impurity 16(R)-5-((3R,5S,6R)-5-amino-6-(2,5-difluorophenyl)tetrahydro-2H-pyran-3-yl)-2-(methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole 5-oxide
MK-3102 Impurity 17N-((2R,3S,5R)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-yl)acetamide
MK-3102 Impurity 18N-((2R,3S,5R)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-yl)benzenesulfonamide
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