乐伐替尼杂质有哪些对照品
深圳远扬化学技术有限公司可提供乐伐替尼项目申报所用全套杂质,随货提供CoA证书,HNMR,MS,HPLC图谱,纯度符合申报要求,现货库存,交货及时,并可根据客户提供结构式进行乐伐替尼杂质定制合成。
乐伐替尼,英文名lenvatinib是一种受体激酶抑制剂,乐伐替尼拥有多个靶点,是一个多靶点靶向药物:VEGFR-1、VEGFR-2、VEGFR-3、FGFR1、PDGFR、cKit、Ret。作为多重靶点的靶向药,乐伐替尼能够透过两个方法阻止癌症细胞的活动:1.抑制肿瘤生成,2.抑制血管形成和过多的生长信号,以达到肿瘤消减。目前被应用于甲状腺癌、肾癌、肝癌等多个癌种。
乐伐替尼属于受体酪氨酸激酶抑制剂,能够阻止血管内皮生长因子受体1 (vascular endothelial growth factorreceptor 1,VEGFR1),VEGFR2以及VEGFR2的激酶活性,抑制新生血管的生成,阻断肿瘤能量的来源从而抑制肿瘤的生长。
乐伐替尼杂质有哪些对照品
乐伐替尼 | CAS号:417716-92-8 | 4-(3-chloro-4-(3-cyclopropylureido)phenoxy)-7-methoxyquinoline-6-carboxamide |
乐伐替尼杂质1 | CAS号:796848-79-8 | 1-(2-chloro-4-hydroxyphenyl)-3-cyclopropylurea |
乐伐替尼杂质2 | CAS号:417721-36-9 | 4-chloro-7-methoxyquinoline-6-carboxamide |
乐伐替尼杂质3 | CAS号:417722-93-1 | 4-(4-amino-3-chlorophenoxy)-7-methoxyquinoline-6-carboxamide |
乐伐替尼杂质4 | CAS号:417717-04-5 | 4-(3-chloro-4-(3-cyclopropylureido)phenoxy)-7-hydroxyquinoline-6-carboxamide |
乐伐替尼杂质5 | CAS号:417717-20-5 | methyl 4-(3-chloro-4-(3-cyclopropylureido)phenoxy)-7-methoxyquinoline-6-carboxylate |
乐伐替尼杂质6 | CAS号:417717-21-6 | 4-(3-chloro-4-(3-cyclopropylureido)phenoxy)-7-methoxyquinoline-6-carboxylic acid |
乐伐替尼杂质7 | CAS号:417714-14-8 | 4-(4-(3-cyclopropylureido)phenoxy)-7-methoxyquinoline-6-carboxamide |
乐伐替尼杂质8 | phenyl (4-((6-carbamoyl-7-methoxyquinolin-4-yl)oxy)-2-chlorophenyl)carbamate | |
乐伐替尼杂质9 | methyl (4-((6-carbamoyl-7-methoxyquinolin-4-yl)oxy)-2-chlorophenyl)carbamate | |
乐伐替尼杂质10 | CAS号:1788901-86-9 | |
乐伐替尼杂质11 | CAS号:417719-45-0 | 4-(3-chloro-4-(3-methylureido)phenoxy)-7-methoxyquinoline-6-carboxamide |
乐伐替尼杂质12 | CAS号:417719-51-8 | 4-(3-chloro-4-ureidophenoxy)-7-methoxyquinoline-6-carboxamide |
乐伐替尼杂质13 | 4-(2-chloro-4-(3-cyclopropylureido)phenoxy)-7-methoxyquinoline-6-carboxamide | |
乐伐替尼杂质14 | 4-(4-amino-3-(4-amino-3-chlorophenoxy)phenoxy)-7-methoxyquinoline-6-carboxamide | |
乐伐替尼杂质15 | 4-(4-((6-carbamoyl-7-methoxyquinolin-4-yl)amino)-3-chlorophenoxy)-7-methoxyquinoline-6-carboxamide |
深圳远扬化学技术有限公司可现货供应各种杂质对照品,医药标准品:阿哌沙班杂质,西曲瑞克杂质,氟替卡松丙酸酯杂质,美沙拉嗪杂质,阿巴卡韦杂质,阿扎胞苷杂质,塞利洛尔杂质,帕瑞昔布杂质,沃替西汀杂质,阿利克仑杂质,地氯雷他定杂质,氟脲嘧啶杂质,美克洛嗪杂质,溴己新杂质,去甲替林杂质,异氟醚杂质,卡维地洛杂质,阿昔洛韦杂质,美克洛嗪杂质,氟康唑杂质,伏立诺他杂质,瑞舒伐他汀杂质,硫酸特布他林杂质,特拉唑嗪杂质,地拉普利杂质,阿戈美拉汀杂质,氯氮平杂质,依匹哌唑杂质,氟伐他汀杂质等,图谱证书齐全,纯度保证。